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YMRF-NH2
目录号:SY-123443
YMRF-NH2为一种神经肽,能特异性结合至FMRFa-R,显示出31 nM的EC50值。
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Ryanodine
目录号:SY-123445
Ryanodine, a diterpenoid poison derived from Ryania speciosa, acts as a modulator of the ryanodine receptor, which is permeable to cells. Depending on its concentration, ryanodine can either stimulate or inhibit Ca2+ release mediated by these receptors.
¥4731.00
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(R)-Lercanidipine-D3 hydrochloride
目录号:SY-123447
(R)-Lercanidipine-D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride (T12626). (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.
¥3312.00
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DL-Phenylalanine-D5
目录号:SY-123449
DL-Phenylalanine-D5是DL-Phenylalanine (TN1592)的氘代物。
¥564.00
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Amlodipine-D4 Maleate (Racemic)
目录号:SY-123451
Amlodipine-D4 Maleate (Racemic)是Amlodipine Maleate (Racemic) (T21263)的氘代化合物。Amlodipine Maleate (Racemic)的CAS号为88150-47-4。Amlodipine maleate是一种具有口服活性的二氢吡啶类钙通道阻滞剂,通过阻滞电压依赖性L型钙通道,从而抑制钙离子内流。Amlodipine maleate可用于研究高血压和癌症。
¥1346.00
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Phenytoin-D10
目录号:SY-123453
Phenytoin-D10 is a deuterated isotope-labelled phenytoin for isotope tracing. Phenytoin (T0939)acts as a voltage-gated Na⁺ channel blocker and t-type Ca²⁺ channel inhibitor,exhibiting antiepileptic activity.
¥2632.00
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Soyacerebroside II
目录号:SY-123455
Soyacerebroside II exhibits ionophoretic activity for Ca2+ ion. Soyacerebrosides I and II have modulating the cellular immune response effects, they show obvious inhibitory activity on IL-18 secretion in human peripheral blood mononuclear cells (PBMC).
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Acetylcholine-D4 chloride
目录号:SY-123457
Acetylcholine-D4 chloride是Acetylcholine chloride (T1221)的氘代物。Acetylcholine chloride (ACh chloride)是一种神经递质,同时也是一种高效的胆碱能 (cholinergic)激动剂。它通过刺激烟碱乙酰胆碱受体 (nAChRs)来调节多巴胺能 (DAergic)神经元的活性。此外,Acetylcholine chloride 能在体外抑制 p53 突变肽的聚集。
¥943.00
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Topiramate-D12
目录号:SY-123459
Topiramate-D12 is a deuterium labeled Topiramate. Topiramate (T0675) is an agent of broad-spectrum antiepileptic. Topiramate (T0675) is an antagonist of GluR5 receptor.
¥2576.00
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