Dynorphin (2-17), amide (porcine)

目录号：SY-112578

Dynorphin (2-17), amide (porcine) 为 dynorphin 衍生物，展现镇痛效果。该化合物源自前体蛋白强啡肽原，涉及阿片肽类，参与疼痛调控、成瘾及情绪调节等生理过程。

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[Nphe1]Nociceptin(1-13)NH2

目录号：SY-112579

Selective and competitive nociceptin receptor antagonist, devoid of any agonist activity. Binds selectively to recombinant nociceptin receptors (pKi = 8.4), and competitively antagonizes the actions of nociceptin in vitro and in vivo.

¥592.00

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Dalargin

目录号：SY-112580

Dalargin 是一种有效的 δ-阿片受体 (δ-opioid receptor) 激动剂。Dalargin 减轻 Gentamicin 诱导的细胞死亡。Dalargin 对庆大霉素诱导的肾损伤具有肾保护作用。Dalargin 具有抗溃疡活性。

¥471.00

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Akuammigine

目录号：SY-112581

Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki val

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Bam 12P

目录号：SY-112582

Bam 12P is a Pro-Met-enkephalin precursor that is isolated from the bovine adrenal medulla.

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β-Endorphin, equine

目录号：SY-112583

Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain. Endorphin Beta is produced in response to pain, exercise, and other forms of stress. Endorphin Beta belongs to a group of

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Nalmefene hydrochloride

目录号：SY-112584

Nalmefene hydrochloride 通过竞争中枢神经系统中的阿片受体来拮抗阿片的作用。

¥760.00

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β-Endorphin (6-31), human

目录号：SY-112585

β-Endorphin是一种内源性阿片类神经肽，作为opioid receptor激动剂，主要与μ-阿片受体发生作用。该肽在中枢和周围神经系统特定神经元中表达，是人类体内三种内啡肽之一。β-Endorphin在减轻压力、维护生理平衡及调控神经系统的疼痛感知中发挥作用。

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Dynorphin A (1-10)

目录号：SY-112586

Dynorphin A (1-10), an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 μM.

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