Ota-vasotocin

目录号：SY-112677

Ota-vasotocin is a ligand utilized in quantitative receptor autoradiography for oxytocin receptors.

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WAY267464 HCl

目录号：SY-112678

WAY267464 is a nonpeptide small-molecule OT agonists with anxiolytic activity. WAY267464 may be used for modulation of potency, selectivity over the structurally similar vasopressin receptors, CNS penetration, and oral bioavailability.

¥4485.00

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(Thr4,Gly7)-Oxytocin

目录号：SY-112679

(Thr4,Gly7)-Oxytocin，一种Oxytocin类似物，特异性激活OT受体。通过激活TRPV1通道及抑制K+通道，诱导眼下神经元兴奋。

¥2850.00

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LIT-001 free base

目录号：SY-112680

LIT-001 free base improves social interaction in a mouse model of autism. LIT-001 free base is the first nonpeptide oxytocin receptor (OT-R) agonist (EC50=55 nM; Ki=226 nM).

¥1725.00

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(Val3,Pro8)-Oxytocin

目录号：SY-112681

"(Val3,Pro8)-Oxytocin"为Gq依赖性途径的激动剂，同时作为β-arrestin结合及催产素受体（OXTR）内化作用的次级激动剂。

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[D-Asn5]-Oxytocin

目录号：SY-112682

[D-Asn5]-Oxytocin exhibits minimal specific oxytocic and vasodepressor effects. Comparative cumulative dose-response investigations reveal that [D-Asn5]-Oxytocin demonstrates a similar intrinsic activity to oxytocin in terms of oxytocic activity.

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JHU-083

目录号：SY-112683

JHU-083 是一种可口服、可穿过血脑屏障且具有选择性的谷氨酰胺酶 (glutaminase) 拮抗剂，可改善 APOE4 小鼠的认知能力，使异常的海马谷氨酰胺酶活性正常化。

¥1881.00

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Nitrosoglutathione

目录号：SY-112684

Nitrosoglutathione (GSNO) 是一种外源性的 NO 供体，是大鼠酒精脱氢酶III 类同工酶的底物，能够减少脑血管紧张素II 依赖性及非依赖型的 AT1 受体反应。

¥180.00

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Sparsentan

目录号：SY-112685

Sparsentan (DARA-a) 是一种具有高度选择的血管紧张素 II (Ki:0.8 nM)和内皮素 A 受体(Ki:9.3 nM)的双重拮抗剂。

¥556.00

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