MK-4541是一种选择性、口服有效的雄激素受体(AR)调节剂，能作为拮抗剂抑制5α-还原酶，从而抑制AR阳性前列腺癌细胞的增殖并诱导凋亡(apoptosis)。此外，MK-4541在异种移植小鼠模型中显著抑制R3327-G前列腺肿瘤的生长。

Cyprodinil 是一种苯胺嘧啶广谱杀菌剂，可抑制植物病原真菌蛋氨酸的生物合成。Cyprodinil 抑制B. cinerea，P. herpotrichoides，H. oryzae 的菌丝体细胞在无氨基酸的培养基上生长，IC50s 分别为 0.44，4.8，0.03 μM。在没有 AR 激动剂 DHT 的情况下，Cyprodinil 充当雄激素受体 (AR) 激动剂 (EC50=1.91 μM)，并抑制 DHT 的雄激素作用 (IC50=15.1 μM)。

non-steroidal androgen receptor (AR) antagonist

11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).

(R)-Bicalutamide 是一种 Bicalutamide 的 R 型对映体，是一种雄激素受体 (AR) 拮抗剂，表现出抗肿瘤效果。(R)-Bicalutamide 广泛的用于前列腺癌的研究。

Leelamine hydrochloride, a tricyclic diterpene extracted from pine tree bark, inhibits the transcriptional activity of the androgen receptor, known to regulate fatty acid synthesis [2,3]. This compound acts as a cannabinoid receptor type 1 (CB1) agonist and suppresses SREBP1-regulated fatty acid/lipid synthesis in prostate cancer cells, irrespective of androgen receptor status.

Dehydroepiandrosterone-d2 是 Dehydroepiandrosterone 的氘代化合物。

Chlormadinone (free base) is a synthetic steroid hormone and antagonist at androgen and estrogen receptors used to treat BPH and polycystic ovary syndrome. It also promotes osteoblast differentiation and Ca deposition in bone marrow stem cells.

Androgen receptor degrader-1 (compound 18)作为高效的雄激素受体降解剂, 主要应用于癌症研究。