LH-RH II (chicken) 为家鸡下丘脑黄体生成素释放激素(LHRH)两种形式之一，亦为哺乳动物LHRH的结构变体。该化合物促进家鸡促性腺激素释放。

Acetyl-ACTH (7-24) (human, bovine, rat) 可导致 ACTH 诱发的皮质酮和醛固酮释放显著减少。

(Rac)-PF-998425 is a potent, selective, nonsteroidal antagonist of the androgen receptor (AR), with IC50 values of 26 nM and 90 nM in AR binding and cellular assays, respectively. This compound shows promise for investigating androgenetic alopecia.

Enzalutamide-d6 (MDV3100-d6) 是氘标记的 Enzalutamide (MDV3100)，一种雄激素受体 (AR) 拮抗剂，在 LNCaP 前列腺细胞中的 IC50为 36 nM。

androgen receptor modulator

ET516 is a strong inhibitor of the Androgen Receptor, effectively halting the proliferation and tumor growth of prostate cancer cells that express AR-resistant mutants [1].

Androgen receptor-IN-6 (compound 16) 是一种口服有效的 Androgen Receptor 抑制剂，具备在体外 IC50=0.12 μM 的效能，专门靶向无序的 N 端结构域 (NTD)。该化合物表现出良好的 Caco2 细胞膜透过性，并在雄性 CD-1 小鼠中展现出 16% 的口服活性 (F/%)。

Androgen receptorligand 3 是雄激素受体 (AR) 配体。通过连接子与 IAP 配体结合，Androgen receptorligand 3 形成 ERαPROTAC 降解剂。

ARCC-4 is an enzalutamide-based von Hippel-Lindau (VHL)-recruiting AR PROTAC and outperforms enzalutamide and it is a low-nanomolar androgen receptor (AR) degrader based on PROTAC, with a DC50 of 5 nM. ARCC-4 effectively degrades clinically relevant AR mutants associated with antiandrogen therapy[1].