Estradiol enanthate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65147，CAS号为 4956-37-0。

Arzoxifene (LY353381) is an orally active selective estrogen receptor modulator (SERM) exhibiting a fixed ring structure analogous to raloxifene. This compound demonstrates potent antiestrogenic effects on breast cancer and endometrium while displaying minimal side effects. Additionally, Arzoxifene elicits favorable estrogenic effects on bone health and lipid profile.

Estrogen receptor-IN-1 (compound 16) 是有效的雌激素受体(ER)抑制剂，其对 ERα 和 Erβ 的IC50值分别为 13 和 5μM。

Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.

Inokosterone is an analgesic drug. It also shows high insect moulting hormone activity.

Imlunestrant (LY-3484356) 是一种口服有效的和选择性的雌激素受体(estrogen receptor)降解剂，能够持续抑制ER依赖基因转录和细胞生长，可用于研究er阳性、her2阴性、esr1突变的晚期或转移性乳腺癌。

Millewanin G shows antiestrogenic activity.

Enclomiphene ((E)-Clomiphene) 是一种有效的、具有口服活性的非甾体雌激素受体 (estrogen receptor) 拮抗剂。Enclomiphene 在睾酮缺乏、男性性腺功能减退症、卵巢功能障碍和 type 2 型糖尿病方面有研究价值。

SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (ERα) ligand 4-hydroxytamoxifen using a PEG linker. It effectively degrades the ERα protein with an IC50 value of 0.097 μM. Within cells, SNIPER(ER)-87 selectively recruits XIAP to ERα, and XIAP functions as the primary E3 ubiquitin ligase responsible for the degradation of ERα induced by SNIPER(ER)-87[1][2].