Bopindolol is a non-selective β-adrenergic receptor antagonist. In vivo, bopindolol decreases heart rate and blood pressure and attenuates ischemia-induced myocardial acidosis in dogs. Formulations containing bopindolol have been used to treat essential and renovascular hypertension.

Cilazapril Monohydrate (Justor) 是一种血管紧张素转化酶抑制剂，能够作用于高血压和充血性心力衰竭的研究。

Aclerastide is an angiotensin receptor agonist. Administration of Aclerastide reduced fibrosis and scarring in the healing wounds. This action was more pronounced with longer administration of the peptide after injury. The action of this peptide was block

(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .

Potent and selective μ opioid receptor antagonist (Ki values are 0.96 and >10,000 nM for μ and δ receptors respectively). Causes behavioral effects on central administration in vivo. Also increases K+ currents in rat locus ceruleus neurons in vitro via a

BNTX (7-Benzylidenenaltrexone) 是选择性δ1-阿片受体拮抗剂。它能竞争性地拮抗 DPDPE、Deltorphin 2 和 DAMGO 的抗分泌功能，并可用于抗伤害作用的研究。

TIPP is an agent of delta opioid antagonist.

Potent, selective partial agonist peptide for the NOP receptor (Ki = 0.71 nM). Selective over μ, δ and κ opioid receptors (IC50 > 4000 nM). Increases food intake in vivo.

[D-Ala2]-Met-Enkephalinamide，一种阿片类肽，有效地作为阿片受体激动剂，通过中枢机制降低胆汁流量并具有镇痛效果。