TLB 150 Benzoate (RAD150) 是一种雄激素受体 (androgen receptor) 的调节剂，其 IC50 值为 0.13 μM。

Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 (NFATc1), this suppression leads to the inhibition of dendritic cell-specific transmembrane pr

Acetyl-ACTH (3-24) (human, bovine, rat) 是原黑色素皮质素 (POMC) 肽的片段。POMC 肽，如促肾上腺皮质激素(ACTH)，是α-MSH 的前体，也是 MC-1 受体的激动剂。

安德罗根受体拮抗剂9（化合物28）作为雄激素受体的对抗物，阻断了该受体的活性。

PROTACAR-V7 degrader-1 (Compound 6)为一种口服有效的，选择性针对AR-V7的降解剂，DC50值为0.32 µM，其作用机制主要是通过VHL E3连接酶将其招募至雄激素受体DNA结合域(AR DBD)。此外，PROTACAR-V7 degrader-1在表达AR-V7的22Rv1细胞系中展现出了活性，EC50值为0.88 µM。

Bromopropylate is an insecticide. Bromopropylate is the active substance in fumigant strips for mites.

Ludaterone is an antiandrogen agent, with potent antiandrogenic activity.

ARCC-4 is an enzalutamide-based von Hippel-Lindau (VHL)-recruiting AR PROTAC and outperforms enzalutamide and it is a low-nanomolar androgen receptor (AR) degrader based on PROTAC, with a DC50 of 5 nM. ARCC-4 effectively degrades clinically relevant AR mutants associated with antiandrogen therapy[1].

Androgen receptorligand 3 是雄激素受体 (AR) 配体。通过连接子与 IAP 配体结合，Androgen receptorligand 3 形成 ERαPROTAC 降解剂。