400-0755-639
联系微信客服
首页 搜索结果
搜索关键词为“”,共搜索43312条结果
Ciwujianoside C1
目录号:SY-127240
Ciwujianoside C1, 一种从Acanthopanax senticosus叶中分离得到的皂苷,具有抑制体外胰腺脂肪酶活性的功能。
¥3312.00
查看详情
Neotheaflavin
目录号:SY-127241
Neotheaflavin, from black tea, inhibits pancreatic lipase.
¥5336.00
查看详情
ERX-41
目录号:SY-127242
ERX-41是一种口服活性的立体特异性小分子,靶向溶酶体酸性脂肪酶A (LIPA)。该化合物通过诱导内质网(ER)应激从而导致细胞死亡,这一作用表明ERX-41功能独立于LIPA,但依赖于其在内质网的定位。ERX-41主要用于实体瘤靶向研究。
¥1035.00
查看详情
(1S)-(+)-Camphor-10-sulphonic acid
目录号:SY-127243
(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。
¥1667.00
查看详情
URB754
目录号:SY-127244
URB754 is a potent and noncompetitive inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 value of 200 nM for the recombinant rat brain enzyme. However, it does not inhibit human recombinant, rat brain, or mouse brain MAGL at concentrations up to 100 μM. There is evidence that the MAGL inhibitory activity of URB754 may be attributed to the impurity bis(methylthio)mercurane (IC50 = 11.9 nM for rat recombinant MAGL) that is found in commercial preparations. URB754 inhibits rat brain fatty acyl amide hydrolase (FAAH) with an IC50 value of 32 μM and binds weakly to the rat central cannabinoid (CB1) receptor with an IC50 value of 3.8 μM. It does not inhibit COX-1 or COX-2 at concentrations up to 100 μM. Inhibition of MAGL hydrolysis of 2-arachidonoyl glycerol (2-AG) is associated with enhanced stress-induced analgesia and may represent a novel drug target in pain and stress management.
¥3312.00
查看详情
PF-06795071
目录号:SY-127245
PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).
¥5336.00
查看详情