Nicardipine is a potent calcium channel blockader with marked vasodilator action.

Lomerizine dihydrochloride (KB-2796) 是一种相对较新的L-和T-型钙通道阻滞剂，用于治疗偏头痛。

Ranolazine (CVT 303, RS 43285-003)是一种钙离子通过 sodium/calcium channal摄取的抑制剂抗心绞痛药物，用于治疗慢性心绞痛。

Ethosuximide(Zarontin)是一种琥珀酰亚胺类的抗痉挛试剂，主要用于失神发作。是钙离子通道阻滞剂。

Sodium tanshinone IIA sulfonate (STS) is a water-soluble derivative of tanshinone IIA isolated as the main pharmacologically active natural compound from a traditional Chinese herbal medicine, the dried root of Salvia miltiorrhiza Bunge known as Danshen. Sodium tanshinone IIA sulfonate (STS) is a potent negative allosteric modulator of the human purinergic receptor P2X7. Sodium tanshinone IIA sulfonate (STS) inhibits the activity of CYP3A4 and store-operated Ca2+ entry (SOCE) through store-operated Ca2+ channels (SOCC) via downregulating the expression of transient receptor potential canonical proteins (TRPC).

Pinaverium bromide (Icosapentaenoic acid)是calcium channel阻滞剂，适用于治疗功能性胃肠病。