PKM2 inhibitor G是丙酮酸激酶抑制剂。

Ophiobolin A is a fungal metabolite and a phytotoxin and is an effective and irreversibly inhibitor of calmodulin-activated cyclic nucleotide phosphodiesterase (IC50: 9 μM). Ophiobolin A also has antimicrobial and anticancer activity.

Metaxalone (Methaxalonum) 具有肌肉松弛作用。

NCGC00188636 (亦称为 DBS) 是一种新型的共价丙酮酸激酶 (PYK) 抑制剂。它通过与丙酮酸激酶的活性位点结合，阻断核苷酸的结合从而抑制酶活性。该化合物展现出对墨西哥乐氏曼原虫丙酮酸激酶 (LmPYK) 的强效抑制作用，可用于研究多种生物及细胞类型的能量代谢过程。

11-Oxoisomogroside V 是从罗汉果(Siraitia grosvenorii)中分离得到的三萜类糖苷化合物，具有抗氧化和抗炎活性。11-Oxoisomogroside V 可激活 PGC-1α 的转录活性。11-Oxoisomogroside V 可提高荧光素酶活性。

4-Nitrophenyl phenylphosphonate is a substrate for 5'-nucleotide phosphodiesterases. It is a more preferable substrate to 5'-nucleotide phosphodiesterases than naturally occurring nucleotides or bis(4-nitrophenyl) phosphate because of its stability, ease of synthesis, and higher rate of hydrolysis under saturating conditions.