Phosphate acceptor peptide

目录号：SY-110081

Phosphate acceptor peptide 是一种 cAMP 依赖性蛋白激酶 (PKA) 的底物。Phosphate acceptor peptide 也是一种弱的PKC 抑制剂。

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PKCd (8-17)

目录号：SY-110080

PKCd (8-17) 是源自蛋白激酶 C (PKC)d V1 结构域的生物活性肽。它能抑制由佛波醇 12-肉豆蔻酸酯 13-乙酸酯 (PMA) 诱导的 PKCd 易位和激活。此外，PKCd (8-17) 在降低心脏和脑细胞缺血损伤、促进成纤维细胞增殖、以及抑制小鼠移植冠状动脉疾病方面具有潜在应用。

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Ilmofosine

目录号：SY-110079

Ilmofosine (BM41440) 是一种高效选择性的蛋白激酶C (protein kinase C) 抑制剂，能够诱导细胞周期在G2期停滞。此外，Ilmofosine 还是一种抗利什曼原虫的药物。

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TLC9995-0188

目录号：SY-110078

Tyrosine-protein kinase ABL, IC50: 1500 nM

¥330.00

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Dihydrosphingosine

目录号：SY-110115

Dihydrosphingosine is a Protein kinase C inhibitor.

¥1694.00

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PKC-theta inhibitor 1

目录号：SY-110114

PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)

¥2442.00

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Bisindolylmaleimide I HCl

目录号：SY-110113

Bisindolylmaleimide I HCl is a specific ATP-competitive PKC inhibitor.

¥363.00

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PKC β pseudosubstrate

目录号：SY-110112

Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia pep

¥2310.00

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(-)-Indolactam V

目录号：SY-110111

(-)-Indolactam V is a PKC activator (Kis: 3.36 nM, 1.03 μM for η-CRD2 , γ-CRD2). (-)-Indolactam V also has the Kds are 5.5 nM (η-C1B), 7.7 nM (ε-C1B), 8.3 nM (δ-C1B), 18.9 nM (β-C1A-long), 20.8 nM (α-C1A-long), 137 nM (β-C1B), 138 nM (γ-C1A), 213 nM (γ-C1

¥1386.00

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