PKM2 activator 4 是PKM2激活剂，AC50值为 1-10 μM。PKM2 activator 4 可用于癌症的研究，

IDO-IN-18是一种强效的吲哚胺 2,3-双加氧酶 (IDO) 抑制剂。它通过阻断色氨酸向犬尿氨酸的转化消除肿瘤微环境的免疫抑制，增强 T 细胞对癌细胞的杀伤活性，常用于癌症免疫治疗研究。

MAO-B-IN-30 是一种可穿过血脑屏障且具有具有选择性和高效性的 MAO-B 抑制剂，具有抗增殖活性，抑制 MAO-A 和 MAO-B 。MAO-B-IN-30 降低 TNF-α、IL-6、NF-kB 在生物体的含量，可用于研究帕金森类的神经系统疾病。

LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.

β-Cembrenediol (β-CBT) is a natural product from tobacco plants that is found in cigarette smoke condensate. β-CBT inhibits induction of the early antigen of Epstein-Barr virus (EA-EBV) by 12-O-tetradecanoylphorbol-13-acetate (TPA) in vitro (IC50 = 21.9 μM). It inhibits tumor promoting effects of TPA on 7,12-demethylbenz[a]anthracene-induced papilloma formation in vivo. β-CBT is also released into soil by flue-cured tobacco plants and exerts autotoxicity as well as phytotoxic activity against L. sativa seedlings.

FCE 28073是一种 Monoamine oxidase B 抑制剂，IC50=0.45 μM。

IDO-IN-7 (NLG-919 analogue) 是 IDO1 抑制剂，IC50=38 nM。

Enpp-1-IN-14 是有效的外核苷酸焦磷酸酶/磷酸二酯酶 (ENPP1) 抑制剂，对重组人 ENPP-1 的 IC50 为 32.38 nM。Enpp-1-IN-14具有抗肿瘤活性。

1,2-Diheptadecanoyl-sn-glycero-3-phosphorylcholine (DHPC) 是生物活性磷脂化合物，属于磷脂酰胆碱 (PC) 的衍生物。