NCGC00188636

目录号：SY-128163

NCGC00188636 (亦称为 DBS) 是一种新型的共价丙酮酸激酶 (PYK) 抑制剂。它通过与丙酮酸激酶的活性位点结合，阻断核苷酸的结合从而抑制酶活性。该化合物展现出对墨西哥乐氏曼原虫丙酮酸激酶 (LmPYK) 的强效抑制作用，可用于研究多种生物及细胞类型的能量代谢过程。

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NPD10084

目录号：SY-128165

NPD10084 是一种靶向丙酮酸激酶 M2 亚型（PKM2）的抑制剂。NPD10084 通过作用于 PKM2 的非糖酵解信号功能，干扰 PKM2 与 β-catenin 或 STAT3 之间的蛋白-蛋白相互作用来抑制下游信号传导，从而对多种结直肠癌细胞系表现出抗增殖活性（体外 IC₅₀范围为 0.8–1.9 μM）。

¥1311.00

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Celgosivir hydrochloride

目录号：SY-126938

Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).

¥9085.00

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Ganoderic acid Y

目录号：SY-126939

Ganoderic acid Y significantly inhibits the replication of the viral RNA (vRNA) of EV71 replication through blocking EV71 uncoating.

¥2530.00

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Prunetin 5-O-β-D-glucopyranoside

目录号：SY-126940

Prunetin 5-O-β-D-glucopyranoside, an isoflavone obtained from Potentilla astracanica extracts, is a potent uncompetitive inhibitor of α-glucosidase (IC 50 = 56.05 μg/mL). It serves as a valuable tool for type-2 diabetes research.

¥6267.00

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2'-Rhamnoechinacoside

目录号：SY-126941

2'-Rhamnoechinacoside is a naturally occurring compound sourced from Cistanche tubulosa.

¥2530.00

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Kouitchenside G

目录号：SY-126942

Kouitchenside G 是一种可以从Swertia kouitchensis 中分离得到的天然产物。Kouitchenside G 抑制α-Glucosidase，IC50为 956 μM。

¥6267.00

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Arisanschinin D

目录号：SY-126943

Arisanschinin D (Ananonin B) 是从 Schisandra arisanensis Hay 中分离的 α-葡萄糖苷酶 (α-Glucosidase) 抑制剂。

¥1438.00

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N-Nonyldeoxynojirimycin

目录号：SY-126944

N-Nonyldeoxynojirimycin (NN-DNJ) is an inhibitor of acid α-glucosidase and α-1,6-glucosidase with IC50 values of 0.42 μM and 8.4 μM, respectively.

¥4600.00

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