PPI-2458 is a synthetic derivative of fumagillin with antineoplastic and cytotoxic properties. PPI-2458 irreversibly inhibits the enzyme methionine aminopeptidase type 2 (MetAP2), thereby preventing abnormal cell growth and angiogenesis. PPI-2458 is reported to have a better toxicity profile compared to other agents of its class.

M8891 is an orally active, reversible and brain penetrant Methionine Aminopeptidase-2 (MetAP-2) inhibitor(IC50 :54nM;Ki:4.33 nM).M8891 inhibits growth of primary endothelial cells as well as tumor cells and demonstrates antiangiogenic and antitumoral acti

4-MDM (4-Methoxydiphenylmethane) 是一种能口服生效的选择性抗炎化合物，通过增强白三烯 A4 水解酶 (LTA4H) 的氨肽酶活性来实现作用。其通过促进LTA4H对脯氨酸-甘氨酸-脯氨酸的降解以减少肺内中性粒细胞的募集，减轻炎症反应，同时不影响LTA4H的环氧水解酶活性。4-MDM 可用于研究与肺部疾病相关的问题。

MetAP2-IN-1为MetAP2抑制剂，用于血管生成介导疾病研究。

TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).

α-Amylase 是一种能够催化淀粉中 α-1,4-糖苷键水解的水解酶，使淀粉产生葡萄糖、麦芽糖等产物。

Docosapentaenoic acid 22n-3 是在所有动物细胞膜中发现的磷脂组成成分。

Ethylidene-4-nitrophenyl-a-D-Maltoheptaoside (pNP-G7) 可作为 α-淀粉酶的底物，用于测量 α-淀粉酶活性。

7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) 可能具有抗真菌c.zeyheri 的作用，是一种潜在的抗真菌药物。它还能抑制药物流出泵(IC50 = 51.64μg /毫升)。