SEA0400 是一种选择性的 Na+-Ca2+ exchanger (NCX) 的强效抑制剂，可抑制神经细胞、星形胶质细胞和小胶质细胞中Na+依赖性的Ca2+吸收，对应的IC50值分别为33 nM、5.0 nM和8.3 nM。SEA0400 可防止硝普钠 (SNP) 提高 ERK 和 p38 MAPK 的磷酸化和通过细胞外Ca2+依赖的方式增强reactive oxygen species (ROS) 的产生。

BIA (TMBIM6 antagonist BIA)是一个潜在的TMBIM6拮抗剂，可以阻断TMBIM6和mTORC2的相互作用，最终阻断AKT的激活和癌症进展。

Ethyl 3-Aminobenzoate (Ethyl m-Aminobenzoate, NSC 93790, Tricaine) 可通过voltage-dependent Na+-channels阻止动作电位的产生，常用于鱼类的麻醉、镇静和安乐死。

BAMB-4 (ITPKA-IN-C14)是一种新型的膜透性的肌醇三磷酸3-激酶A(Inositol-Trisphosphate 3-Kinase A, ITPKA)抑制剂，在ADP-Glo激酶检测中，IC50为37 μM。

Rhynchophylline (Mitrinermine), an active component isolated from species of the genus Uncaria, acts as a calcium channel blocker and is widely used in traditional Chinese medicine mainly for treating ailments of central nervous and cardiovascular systems, such as lightheadedness, convulsions, numbness, and hypertension.

Z944是一种高度选择性的T型钙通道拮抗剂，对hCaV3.1、hCaV3.2和hCaV3.3的IC50分别为50、160、110 nM。

Protopine (Corydinine, Fumarine, Biflorine, Macleyine), an alkaloid present in different plants, has been shown to exhibit a number of activities, such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation. It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities.

Azumolene（EU4093 free base）是一种等效的丹曲林（dantrolene）类似物，是一种兰尼碱受体 (ryanodine receptor, RyR) 调节剂，可抑制钙释放。