(E)-4-Hydroxytamoxifen

目录号：SY-111964

(E)-4-Hydroxytamoxifen is a less active isomer of (Z)-4-hydroxytamoxifen and also is an estrogen receptor modulator.

¥583.00

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Raloxifene 4-Monomethyl Ether

目录号：SY-111965

Raloxifene 4-Monomethyl Ether (Compound 37) is a derivative of Raloxifene which acts as an inhibitor of estrogen receptor α. It effectively suppresses the activity of MCF-7 cells, exhibiting an IC50 value of 1 μM and a pIC50 value of 6.

¥3323.00

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Bexirestrant

目录号：SY-111966

Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.

¥4174.00

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ZK 164015

目录号：SY-111967

estrogen receptor silent antagonist

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Dienestrol diacetate

目录号：SY-111968

Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activities.

¥240.00

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Benzophenone-2

目录号：SY-111969

Benzophenone-2 (2,2',4,4'-Tetrahydroxybenzophenone) 是一种内分泌干扰物，主要靶向孕烷 X 受体 (PXR) 和雌激素受体 α (ERα)。通过激活 PXR，Benzophenone-2 能够调节细胞色素 P450 3A (CYP3A) 的表达。该化合物有潜力在紫外线过滤剂的研究中得到应用。

¥32.00

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PROTAC ER Degrader-4

目录号：SY-111970

PROTAC ER Degrader-4 is a PROTAC degrader of the estrogen receptor (ER) with an IC50 of 0.8 nM.

¥2750.00

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ERD-308

目录号：SY-111971

ERD-308 induces >95% of ER degradation at concentrations as low as 5 nM in both cell lines (DC50 (concentration causing 50% of protein degradation) of 0.17 nM and 0.43 nM in MCF-7 and T47D ER+ cells, respectively).ERD-308 is a highly potent PROTAC degrade

¥1056.00

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Enclomiphene hydrochloride

目录号：SY-111972

Enclomiphene ((E)-Clomiphene) hydrochloride 是一种口服具有活力的、有效的非甾体雌激素受体 (estrogen receptor) 拮抗剂，具有抗雌激素作用。Enclomiphene hydrochloride 能够用于研究卵巢功能障碍、睾酮缺乏、男性性腺功能减退症和 type 2 型糖尿病。

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