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Acetylcholine-D4 bromide
目录号:SY-123375
Acetylcholine-D4 bromide是Acetylcholine bromide (T20344)的氘代形式。
¥471.00
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L-Phenylalanine-13C9,15N
目录号:SY-123417
L-Phenylalanine-13C9,15N是经过 13C 和 15N 标记的 L-Phenylalanine (T3377)。L-Phenylalanine ( (S)-2-Amino-3-phenylpropionic acid)是一种从大肠杆菌中提取的必需氨基酸。它作为电压依赖性 α2δ 亚基 Ca2+ 通道的拮抗剂,Ki 值为 980 nM,并且是NMDARs (KB 573 μM)和非 NMDARs 之中甘氨酸和谷氨酸结合点的竞争性拮抗剂。L-Phenylalanine 还广泛应用于食品香料和药物的制造。
¥1782.00
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4-Bromo A23187
目录号:SY-123395
4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.
¥1925.00
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Ryanodine
目录号:SY-123445
Ryanodine, a diterpenoid poison derived from Ryania speciosa, acts as a modulator of the ryanodine receptor, which is permeable to cells. Depending on its concentration, ryanodine can either stimulate or inhibit Ca2+ release mediated by these receptors.
¥4731.00
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Acetylcholine-D4 chloride
目录号:SY-123457
Acetylcholine-D4 chloride是Acetylcholine chloride (T1221)的氘代物。Acetylcholine chloride (ACh chloride)是一种神经递质,同时也是一种高效的胆碱能 (cholinergic)激动剂。它通过刺激烟碱乙酰胆碱受体 (nAChRs)来调节多巴胺能 (DAergic)神经元的活性。此外,Acetylcholine chloride 能在体外抑制 p53 突变肽的聚集。
¥943.00
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Praziquantel
目录号:SY-123211
Praziquantel (Droncit) 是一种外消旋混合物,由 (R)-Praziquantel 和 (S)-Praziquantel 组成。它可研究血吸虫病。
¥88.00
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ABT-639
目录号:SY-123181
ABT-639 是一种有效的选择性 T 型钙通道阻滞剂。
¥462.00
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Gallopamil
目录号:SY-123209
Gallopamil (Methoxyverapamil) 是一种苯烷基胺钙拮抗剂,以浓度依赖性方式抑制酸分泌 (IC50 = 10.9 μM)。Gallopamil 显示出抗心律失常和血管扩张剂的功效。
¥299.00
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Phenytoin-D10
目录号:SY-123453
Phenytoin-D10 is a deuterated isotope-labelled phenytoin for isotope tracing. Phenytoin (T0939)acts as a voltage-gated Na⁺ channel blocker and t-type Ca²⁺ channel inhibitor,exhibiting antiepileptic activity.
¥2632.00
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