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GPR35 agonist 1
目录号:SY-112261
GPR35 agonist 1 is a highly effective and specific GPR35/CXCR8 agonist (EC50: 5.8 nM).
¥2464.00
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Commendamide
目录号:SY-112265
Commendamide is a natural bacterial product that was discovered in a screen for commensal bacteria effector genes (Cbegs). Cbeg12 is a bacterial effector gene that encodes for its production. Commendamide is structurally similar to long-chain N-acyl-amides, which commonly signal, in mammals, through G protein-coupled receptors. Commendamide activates GPR132 (also known as G2A) with an EC50 value of 11.8 μM.
¥1518.00
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ATC0065 HCl
目录号:SY-112269
ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.
¥1610.00
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Melanin Concentrating Hormone, salmon
目录号:SY-112273
Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.
¥2288.00
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Monomethyl fumarate-d3
目录号:SY-112277
Monomethyl fumarate D3 is a deuterium labeled Monomethyl fumarate.
¥1414.00
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Miricorilant
目录号:SY-112281
Miricorilant (CORT 118335) 是一种选择性糖皮质激素受体调节剂,可用于研究消化系统疾病和代谢疾病。
¥2277.00
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Spirorenone
目录号:SY-112285
Spirorenone (INN)是一种新型醛固酮拮抗剂,具有抗盐皮质激素活性,可用于研究代谢疾病。
¥3024.00
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Prednisone acetate
目录号:SY-112289
Prednisone acetate (Prednisone 21-acetate) 是泼尼松的醋酸盐形式,它是一种糖皮质激素受体激动剂,具有抗炎和免疫调节作用。
¥475.00
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SCO-267
目录号:SY-112194
SCO-267是一种GPR40/FFAR1完全激动剂,EC50=12 nM,有效刺激糖尿病大鼠胰岛素分泌和GLP-1释放,改善糖耐量,可用于治疗2型糖尿病。
¥432.00
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