(R)-6',7'-Dihydroxybergamottin is an ihhibitor of CYP1A1 and the isomer of 6',7'-Dihydroxybergamottin(DHB).

Isavuconazole-D4 Isavuconazole (T2305)D4 is a deuterium labeled Isavuconazole. Isavuconazole (T2305) is a triazole prodrug with antifungal activity against yeasts,molds,and dimorphic fungi.

Tebuconazole-D9 is intended for use as an internal standard for the quantification of tebuconazole by GC- or LC-MS. Tebuconazole (T17022) is a triazole fungicide that is active against both seed and foliar fungi. It inhibits 14α-demethylase isolated from U. maydis and S. bicolor with IC50 values of 0.05 and 0.16 nM,respectively. It inhibits the androgenic effect of the androgen receptor agonist DHT (IC20 = 2.89 µM)and is cytotoxic (EC20 = 38.9 µM)in an MDA-kb2 assay. Tebuconazole (T17022) (50 and 100 mg/kg per day)administered during gestation reduces testosterone levels and increases testicular levels of progesterone and 17α-hydroxyprogesterone in male rat fetuses. It has a feminizing effect on male pups and a virializing effect on female pups. When administered to rats gestationally through postnatal day 42,tebuconazole (20 and 60 mg/kg per day)leads to cell death of pyramidal cells in the CA3-4 region of the hippocampus and layer V of the cortex concomitant with impairment in learni

Dasatinib Analog-1，其Ki值为5.4 μM，能够抑制CYP3A4活力，并能阻断谷胱甘肽加合物的形成。

EMT inhibitor-2 inhibits CYP3A4 testosteron and CYP2C9 with IC50s of 49.72 and 5.54 μM, respectively. EMT inhibitor-2 inhibits epithelial-mesenchymal transition (EMT) induced by substances such as IL-1β and TGF-β released from the immunocytes.

(4S,5S)-(+)-Germacrone-4,5-epoxide inhibits certain subtypes of cytochrome P450 (CYP).