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Imatinib Impurity E
目录号:SY-124271
Imatinib Impurity E 是 Imatinib 的杂质。Imatinib 是一种口服生物可用的酪氨酸激酶抑制剂,可选择性抑制 BCR/ABL,v-Abl,PDGFR,c-kit 激酶活性。Imatinib (STI571) 靠近 ATP 结合位点结合,将其锁定在封闭或自我抑制的构象中,因此半竞争性抑制蛋白质的酶活性。Imatinib 还抑制 SARS-CoV 和MERS-CoV。
¥1276.00
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Methyl 2,4,6-trihydroxybenzoate
目录号:SY-124273
Methyl 2,4,6-trihydroxybenzoate 是 2,4,6-trihydroxybenzoate 的代谢产物,可从洋葱皮中分离得到,具有抗氧化、降脂和抗癌活性。Methyl 2,4,6-trihydroxybenzoate 通过氢原子转移(HAT)与单电子转移(SET)清除自由基(DPPH・、ABTS・⁺、・OH),抑制脂质过氧化。Methyl 2,4,6-trihydroxybenzoate可用于抗肿瘤研究。
¥425.00
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3-Oxo Atorvastatin
目录号:SY-124274
3-Oxo Atorvastatin, an impurity of Atorvastatin, acts as an HMG-CoA reductase inhibitor and effectively decreases blood lipids.
询价
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Iloperidone metabolite Hydroxy Iloperidone
目录号:SY-124275
Iloperidone metabolite Hydroxy Iloperidone is an atypical antipsychotic. It is a metabolite of Iloperidone.
¥1539.00
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6-Hydroxybentazon
目录号:SY-124276
6-Hydroxybentazon is a phase I metabolite of bentazon, a herbicide.
¥1035.00
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Tofacitinib metabolite-1
目录号:SY-124277
Tofacitinib metabolite-1, a derivative of Tofacitinib, which is a JAK inhibitor, is employed in studies focused on the pharmacokinetics and metabolism of tofacitinib[1][2].
¥966.00
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