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Amlodipine aspartic acid impurity
目录号:SY-123406
Amlodipine aspartic acid is a calcium channel blocker compound that exhibits antihypertensive and antianginal properties. It is important to note that Amlodipine aspartic acid impurity is an impurity specific to this compound.
¥805.00
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L-Phenylalanine-13C9,15N,D8
目录号:SY-123408
L-Phenylalanine-13C9,15N,D8是一种带有13C,15N 标记和氘代标记的L-Phenylalanine (T3377)。L-Phenylalanine ( (S)-2-Amino-3-phenylpropionic acid)是从大肠杆菌中分离出来的必需氨基酸。它是一种电压依赖性α2δ亚基Ca2+通道拮抗剂,Ki值为980 nM。L-Phenylalanine 还是NMDARs (KB573 μM)和非NMDARs的甘氨酸和谷氨酸结合位点的竞争性拮抗剂,广泛用于食品香料和药品的生产。
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Adenophostin A
目录号:SY-123410
Adenophostin A 是一种高效的肌醇三磷酸 (IP3) 受体激动剂,它能与IP3受体高亲和力结合,促进钙离子 (Ca2+) 的释放。
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Zeorin
目录号:SY-123412
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24-BSA, it shows potent inhibitory effect by 40% decrease of histamine release.
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Cimicifugic acid D
目录号:SY-123414
Cimicifugic acid D (2-Caffeoylpiscidic acid) 是一种苄基酒石酸酯,能够诱导预收缩的大鼠主动脉条血管扩张,并启动内皮依赖性舒张机制。在Norepinephrine引起的大鼠主动脉条收缩过程中,Cimicifugic acid D 通过抑制受体操纵的Ca2+通道(ROC)的胞外Ca2+内流发挥作用,而不影响电压依赖性Ca2+通道(VDC)或K+诱导的收缩。
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L-Phenylalanine-13C
目录号:SY-123416
L-Phenylalanine-13C是一种具有 13C 标记的 L-Phenylalanine (T3377)。L-Phenylalanine ( (S)-2-Amino-3-phenylpropionic acid)是从大肠杆菌中提取的必需氨基酸,作为电压依赖性 α2δ 亚基 Ca2+ 通道的拮抗剂,其 Ki 为 980 nM。此外,L-Phenylalanine是NMDARs (Kᵦ 573 μM)和非NMDARs 甘氨酸和谷氨酸结合位点的竞争性拮抗剂,广泛应用于食品香料和药品的制造。
¥575.00
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