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IYPTNGYTR
目录号:SY-124474
IYPTNGYTR, a deamidation-sensitive peptide, is a deamidation derivative of Trastuzumab. This compound, IYPTNGYTR, can be utilized for monitoring Trastuzumab metabolism in vivo.
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4-Desmethoxy Omeprazole
目录号:SY-124179
4-Desmethoxy Omeprazole 是 Omeprazole 的活性代谢物。Omeprazole 是质子泵抑制剂。Omeprazole 竞争性抑制 CYP2C19 活性,Ki=2 - 6 μM。Omeprazole 还抑制革兰氏阴性菌和革兰氏阳性菌生长。
¥736.00
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Vanillylmandelic acid
目录号:SY-125067
Vanillylmandelic acid 是儿茶酚胺、肾上腺素和去甲肾上腺素代谢的最终产物,具有抗氧化活性,常用于帮助诊断嗜铬细胞瘤,以及其升高与抑郁症状有关。
¥264.00
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Anselamimab
目录号:SY-123124
Anselamimab(安赛埃单抗)是一种人源化IgG1κ单克隆抗体,靶向血清淀粉样蛋白A1(SAA1)。它通过特异性结合淀粉样纤维,触发巨噬细胞和中性粒细胞的吞噬作用,从而清除淀粉样沉积物。Anselamimab在临床期中作为APP抑制剂((β-amyloid A4 Protein Precursor),用于治疗轻链(AL)淀粉样变性。
¥2277.00
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Isavuconazole-D4
目录号:SY-123726
Isavuconazole-D4 Isavuconazole (T2305)D4 is a deuterium labeled Isavuconazole. Isavuconazole (T2305) is a triazole prodrug with antifungal activity against yeasts,molds,and dimorphic fungi.
¥2369.00
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Permethric acid
目录号:SY-124383
Permethric acid 是杀虫剂氯菊酯(permethrin)的代谢物。
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N-desmethylmirtazapine
目录号:SY-124093
N-desmethylmirtazapine (J1.061.658A) 是mirtazapine 的代谢物。它也常用作抗焦虑药、催眠药、止吐药和食欲兴奋剂。
¥897.00
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Nampt-IN-5
目录号:SY-123612
Nampt-IN-5 是烟酰胺磷酸核糖基转移酶抑制剂。它可抑制 A2780 和 COR-L23 细胞,IC50值分别为 0.7 nM 和 3.9 nM。它还抑制 CYP3A4 活性。
¥702.00
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TFM
目录号:SY-123760
TFM is a piscicide.1It is toxic to sea lamprey (P. marinus) with LC50values ranging from 1.97 to 2.11 and 2.05 to 2.21 mg/L for sac and swim-up fry, respectively, 1.6 to 2.45 mg/L for juveniles, and 1.6 to 1.63 mg/L for adults. It is also toxic to juvenile lake sturgeon (A. fulvescens) less than 100 mm in size but not to a variety of other fish species. TFM (50 μM) uncouples oxidative phosphorylation by 22 and 28% in isolated sea lamprey and rainbow trout (O. mykiss) liver, respectively.2Formulations containing TFM have been used as lampricides in the control of larval sea lamprey populations. 1.Boogaard, M.A., Bills, T.D., and Johnson, D.A.Acute toxicity of TFM and a TFM/niclosamide mixture to selected species of fish, including lake sturgeon (Acipenser fulvescens) and mudpuppies (Necturus maculosus), in laboratory and field exposuresJ. Great Lakes Res.29(Suppl 1)529-541(2003) 2.Birceanu, O., McClelland, G.B., Wang, Y.S., et al.The lampricide 3-trifluoromethyl-4-nitrophenol (TFM) unco
¥115.00
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