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Imperatoxin A
目录号:SY-123315
Imperatoxin A,源自非洲蝎Pandinus imperator毒液的一种肽毒素,作为Ca2+-释放通道/兰尼碱受体(RyRs)的激活剂,促进Ca2+从肌浆网流入细胞。
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Vindorosine
目录号:SY-123319
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular smooth muscles.
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Aprindine hydrochloride
目录号:SY-123307
Aprindine HCl is a Class 1b antiarrhythmic agent used to manage ventricular and supraventricular arrhythmias. In one study, it delayed atrial fibrillation more than digoxin did. It has shown effectiveness when given orally.
¥770.00
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piCRAC-1
目录号:SY-123393
piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel. It effectively alleviates thrombocytopenia and hemorrhage [1].
¥1606.00
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ω-Conotoxin GVIA
目录号:SY-123385
Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.
¥2656.00
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ABT-639
目录号:SY-123181
ABT-639 是一种有效的选择性 T 型钙通道阻滞剂。
¥462.00
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IDO1-IN-19
目录号:SY-123461
IDO1-IN-19 (Compound 17) 是一种 IDO1 的有效抑制剂,具有潜力进行癌症疾病的研究。
¥737.00
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HSK16149
目录号:SY-123301
HSK16149 是一种新型的电压门控钙离子通道(VGCC)α2δ亚基选择性配体,具有镇痛活性。
¥3910.00
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KT-362 fumarate
目录号:SY-123156
KT-362 fumarate 是一种新型化合物,可作为钙通道、钾通道和钠通道的拮抗剂.KT-362 fumarate 通过影响心房肌肉细胞内钙动员导致血管舒张。KT-362 fumarate 对兔子的股动脉和基底动脉条有放松作用。
¥2599.00
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