400-0755-639
联系微信客服
最新产品
三叶新科每月上新,持续为科研人员提供新颖性研究工具,助力科研创新与突破。
首页 最新产品
MB-07803
目录号:SY-128271
MB07803 is an orally available prodrug of an effective, noncompetitive inhibitor of fructose 1,6-bisphosphatase (FBPase) (EC50: 140 nM and t1/2 of 7.6±2.9 h).This compound is unstable in powder form and other related salt forms are recommended.
询价
查看详情
Calyculin A
目录号:SY-128266
Calyculin A ((-)-Calyculin A) 是日本海洋海绵 CDiscodermia calyxC 中的毒性物质,是一种具有选择性和高效性的蛋白磷酸酶 1 (PP1) 和蛋白磷酸酶 2A (PP2A) 抑制剂, 诱导冷冻保存牛精子的过度激活,抑制人淋巴细胞中辐射诱导的 gammaH2AX DNA 修复病灶的消失。
¥10450.00
查看详情
2-Bromo-4'-hydroxyacetophenone
目录号:SY-128257
2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) 是一种PTP1B 的有效抑制剂,其Ki=42 μM。
¥95.00
查看详情
ARL-67156 trisodium salt hydrate
目录号:SY-128285
ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.
询价
查看详情
PPM1A-IN-1
目录号:SY-128289
PPM1A-IN-1(Compound IV-4)是一种小分子抑制剂,可特异性抑制 Mg²⁺/Mn²⁺ 依赖的蛋白磷酸酶 PP2C Ser/Thr phosphatase 1A。通过干扰关键去磷酸化过程,PPM1A-IN-1 对结核分枝杆菌表现出显著的抗菌活性,广泛用于抗结核药物开发及磷酸酶靶点机制研究。
询价
查看详情
AQX-435
目录号:SY-128287
AQX-435 是一种有效的 SHIP1 (SH2 domain-containing inositol-5′-phosphatase 1) 激活剂。AQX-435 能够降低 B 细胞受体 (BCR) 下游 PI3K 活性,诱导恶性 B 细胞凋亡,对淋巴瘤生长表现出抑制作用。
¥5775.00
查看详情
MY33-3
目录号:SY-128275
MY33-3 is a powerful and specific inhibitor of receptor protein tyrosine phosphatase (RPTP)β/ζ, demonstrating an IC50 value of approximately 0.1 μM. Moreover, MY33-3 exhibits inhibitory activity against PTP-1B with an IC50 value of about 0.7 μM. Additionally, MY33-3 has been shown to effectively decrease ethanol consumption and alleviate neuroinflammation and cognitive dysfunction induced by Sevoflurane.
询价
查看详情
2-Hydroxy-3-(hydroxymethyl)anthraquinone
目录号:SY-128284
2-Hydroxy-3-(hydroxymethyl)anthraquinone 在 Hepa lclc7 细胞中表现出醌还原酶 (QR) 诱导活性,其 QR 活性加倍所需的浓度为 0.94 microM。
询价
查看详情
Rhein-8-glucoside calcium
目录号:SY-128269
Rhein-8-glucoside calcium (Rhein-8-glucoside calcium salt) salt 是一种从 Saussurea lappa 根的 EtOH 提取物中,分离得到的蒽醌类 hPTP1B 抑制剂,IC50值为11.5 μM,具有抗菌作用。
¥5130.00
查看详情