LKY-047, a derivative of Decursin, is a highly effective and specific reversible competitive inhibitor of cytochrome P45022J2 (CYP2J2), with an IC 50 value of 1.7 μM. LKY-047 does not display inhibitory activity against other human P450 enzymes including CYPs 1A2, 2A6, 2B6, 2C8, 2C9, 2C19, 2D6, 2E1, and 3A.

5,6,7-Trimethoxycoumarin shows moderate inhibitory activity against Micrococcus luteus, it also displays an intermediate cytotoxic effects against brine shrimp larvae. 5,6,7-Trimethoxycoumarin can improve gastroprotective effects, and it has low toxicity

Atazanavir-D6是Atazanavir (T0100L)的氘代化合物。Atazanavir的CAS号为198904-31-3。Atazanavir是一种高选择性的HIV-1蛋白酶抑制剂，可研究艾滋病毒感染。它也是SARS-CoV 3CLpro的抑制剂，IC50为 3.49 μM。它是CYP3A4的底物和抑制剂，也是P-糖蛋白的抑制剂和诱导剂。

Quilseconazole is an effective, orally active fungal Cyp51 inhibitor. it also binds tightly to cryptococcal CYP51 but weakly inhibits humans CYP450 enzymes.

2',5,6',7-Tetrahydroxyflavone 是一种从植物中分离到的黄酮类天然产物。

3-Phenylthiophene (Compound 25) 是一种CYP2A6抑制剂，Ki值为3.3 μM。其对CYP2E1、CYP2B6、CYP2C9、CYP2C19的Ki分别为9.7、14、112和107 μM，对CYP3A4和CYP2D6无显著抑制作用，可用于戒烟研究。