Bepridil hydrochloride (CERM 1978) 是一种钙通道阻滞剂，还抑制 Na+/Ca2+ 交换(NCX)、钠通道和心脏肌膜 KATP 通道，具有抗心绞痛的作用。

Gabapentin-D4是Gabapentin (T0702)的氘代化合物。Gabapentin的CAS号为60142-96-3。Gabapentin是GABA类似物，是一种抗癫痫药，可用于缓解神经性疼痛。

(S)-Lercanidipine-D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride (T12804) is an agent of antihypertensive.

Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂，可抑制放射性配体与毒蕈碱 M1 结合。

Fukinolic acid 是一种苄基酒石酸酯，作为血管扩张剂，显示出抑制肠道病毒A71 (EV-A71) 复制的效果。它是受体调控的Ca2+通道 (ROC) 的抑制剂，通过抑制 Norepinephrine 激活的 ROC 来阻止细胞外Ca2+ 的内流，而不影响电压依赖性Ca2+通道。

TMB 8 is a non-competitive antagonist of nicotinic acetylcholine receptors (nAChRs) with IC50 values of 390 and 350 nM, respectively, for human muscle-type and α3β4 subunit-containing ganglionic nAChRs expressed in TE671/RD or SH-SY5Y cells. It inhibits nicotine-induced dopamine release from rat brain synaptosomes (IC50 = 480 nM). TMB 8 also reduces calcium availability in smooth and skeletal muscle, blocking the contractile response in isolated rabbit aortic strip when used at a concentration of 50 μM and inhibiting calcium influx and efflux in isolated guinea pig ileum when used at a concentration of 65 μM. It has been used in the study of intracellular calcium dynamics, particularly in smooth muscle. TMB 8 also inhibits protein kinase C (PKC) activity in a dose-dependent manner.

ω-Conotoxin SVIB为从Conus venoms中分离得到的肽类毒素，具有抑制抽搐反应的能力，IC50值为37 nM。在小鼠体内，ω-Conotoxin SVIB可导致呼吸急迫，并在高浓度下致死。

L-Phenylalanine-13C是一种具有 13C 标记的 L-Phenylalanine (T3377)。L-Phenylalanine ( (S)-2-Amino-3-phenylpropionic acid)是从大肠杆菌中提取的必需氨基酸，作为电压依赖性 α2δ 亚基 Ca2+ 通道的拮抗剂，其 Ki 为 980 nM。此外，L-Phenylalanine是NMDARs (Kᵦ 573 μM)和非NMDARs 甘氨酸和谷氨酸结合位点的竞争性拮抗剂，广泛应用于食品香料和药品的制造。

Isokaempferide shows hepatoprotective, antiproliferative, and anti-inflammatory effects, the anti-inflammatory effects can be explained, at least in part, by reducing neutrophil degranulation, myeloperoxidase activity, mediators as well as TNF-alpha secretion. Isokaempferide is used as a bronchodilator, can induce relaxation of guinea-pig isolated trachea.